- Class: 1
- Architecture: 1.10:Orthogonal Bundle
- Topology: 1.10.287:Helix Hairpins
- Homology: 1.10.287.940:atp-gated p2x4 ion channel
PDB Entries
PDB ID | OPM | Mutant | Chain Formula | Resolution | HETNAM | |||
---|---|---|---|---|---|---|---|---|
Amino Acid sequence | SCOPe Family Level | CATH Homology Level | ||||||
3h9v | [A3] | [A3] | [A3] | 3.1 | GD:GADOLINIUM ATOM NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
3i5d | [A3] | [A3] | [A3] | 3.46 | NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
4dw0 | [A3] | [A3] | [A3] | 2.9 | BMA:BETA-D-MANNOPYRANOSE GD:GADOLINIUM ATOM GOL:GLYCEROL MAN:ALPHA-D-MANNOPYRANOSE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
4dw1 | [A3] | [A3] | [A3] | 2.8 | ATP:ADENOSINE-5___sq___-TRIPHOSPHATE BMA:BETA-D-MANNOPYRANOSE GOL:GLYCEROL MAN:ALPHA-D-MANNOPYRANOSE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5f1c | [A3] | [A3] | [A3] | 2.9 | ATP:ADENOSINE-5___sq___-TRIPHOSPHATE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE ZN:ZINC ION | |||
5svj | [A3] | [A3] | [A3] | 2.98 | EDO:1,2-ETHANEDIOL MG:MAGNESIUM ION NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE PG4:TETRAETHYLENE GLYCOL | |||
5svl | [A3] | [A3] | [A3] | 2.9 | ACT:ACETATE ION ATP:ADENOSINE-5___sq___-TRIPHOSPHATE EDO:1,2-ETHANEDIOL GLC:ALPHA-D-GLUCOPYRANOSE NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE TRS:2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL | |||
5svm | [A3] | [A3] | [A3] | 3.09 | 6AT:2-(METHYLSULFANYL)ADENOSINE 5___sq___-(TETRAHYDROGENTRIPHOSPHATE) ATP:ADENOSINE-5___sq___-TRIPHOSPHATE EDO:1,2-ETHANEDIOL NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE TRS:2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL | |||
5svp | [A3] | [A3] | [A3] | 3.3 | 6AT:2-(METHYLSULFANYL)ADENOSINE 5___sq___-(TETRAHYDROGENTRIPHOSPHATE) ATP:ADENOSINE-5___sq___-TRIPHOSPHATE EDO:1,2-ETHANEDIOL NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE TRS:2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL | |||
5svq | [A3] | [A3] | [A3] | 3.25 | 128:SPIRO(2,4,6-TRINITROBENZENE[1,2A]-2O___sq___,3O___sq___-METHYLENE-ADENINE-TRIPHOSPHATE MG:MAGNESIUM ION NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5svr | [A3] | [A3] | [A3] | 3.13 | 71C:5-{[(3-PHENOXYPHENYL)METHYL][(1S)-1,2,3,4-TETRAHYDRONAPHTHALEN-1-YL]CARBAMOYL}BENZENE-1,2,4-TRICARBOXYLIC ACID MG:MAGNESIUM ION NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5svt | [A3] | [A3] | [A3] | 3.79 | MG:MAGNESIUM ION NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1l | [A3] | [A3] | [A3] | 3.4 | NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1u | [A3] | [A3] | [A3] | 3.6 | 7S4:N-{(1R)-1-[N___sq______sq___-CYANO-N___sq___-(QUINOLIN-5-YL)CARBAMIMIDAMIDO]-2,2-DIMETHYLPROPYL}-2-(3,4-DIMETHOXYPHENYL)ACETAMIDE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1v | [A3] | [A3] | [A3] | 3.4 | 7S1:N-CYANO-N___sq___-[(1R)-1-PHENYLETHYL]-N___sq______sq___-QUINOLIN-5-YLGUANIDINE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1w | [A3] | [A3] | [A3] | 3.5 | 7RY:N-[2-({2-[(2-HYDROXYETHYL)AMINO]ETHYL}AMINO)QUINOLIN-5-YL]-2-[(3S,5S,7S)-TRICYCLO[3.3.1.1~3,7~]DECAN-1-YL]ACETAMIDE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1x | [A3] | [A3] | [A3] | 3.2 | 7RV:N-{[4-(4-PHENYLPIPERAZIN-1-YL)OXAN-4-YL]METHYL}-2-(PHENYLSULFANYL)PYRIDINE-3-CARBOXAMIDE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u1y | [A3] | [A3] | [A3] | 3.3 | 7RS:N~2~-(3,4-DIFLUOROPHENYL)-N-{2-METHYL-5-[(PIPERAZIN-1-YL)METHYL]PHENYL}GLYCINAMIDE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5u2h | [A3] | [A3] | [A3] | 3.9 | 7S1:N-CYANO-N___sq___-[(1R)-1-PHENYLETHYL]-N___sq______sq___-QUINOLIN-5-YLGUANIDINE ATP:ADENOSINE-5___sq___-TRIPHOSPHATE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5wzy | [A3] | [A3] | [A3] | 2.8 | BMA:BETA-D-MANNOPYRANOSE CTP:CYTIDINE-5___sq___-TRIPHOSPHATE GOL:GLYCEROL MAN:ALPHA-D-MANNOPYRANOSE NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE | |||
5yve | [A3] | [A3] | [A3] | 3.4 | AF9:5-[2,4-BIS(AZANYL)PYRIMIDIN-5-YL]OXY-2-METHOXY-4-PROPAN-2-YL-BENZENESULFONAMIDE MG:MAGNESIUM ION NA:SODIUM ION NAG:2-ACETAMIDO-2-DEOXY-BETA-D-GLUCOPYRANOSE |
*Chain Formula of OLIGAMI.
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA
[ ] : Polypeptide - [AB] : Protein, [ab] : Small peptide
( ) : Nucleic acid - (AB) : DNA, (ab) : RNA